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Volume 9
Main Index

Issue 1


Synthesis and Pharmacology of 6-Methylenedihydrodesoxymorphine
M. Adawi Abdel-Rahman, Henry W. Elliott, Robert Binks, Werner Küng, and Henry Rapoport
pp 1 - 6; DOI:
10.1021/jm00319a001
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Analgesic Antagonists. I. 4-Substituted 1-Acyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepines
P. M. Carabateas and L. S. Harris
pp 6 - 10; DOI:
10.1021/jm00319a002
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Thyromimetics. V. The Synthesis and Biological Screening of α-Methylthyroxine
Benjamin Blank, Edward G. Rice, Francis R. Pfeiffer, and Cyrus M. Greenberg
pp 10 - 15; DOI:
10.1021/jm00319a003
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Fusidic Acid Derivatives. I. Relationship between Structure and Antibacterial Activity
W. O. Godtfredsen, W. von Daehne, L. Tybring, and S. Vangedal
pp 15 - 22; DOI:
10.1021/jm00319a004
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Biologically Active Guanidines and Related Compounds. II. Some Antiinflammatory Aminoguanidines
G. J. Durant, G. M. Smith, R. G. W. Spickett, and S. H. B. Wright
pp 22 - 27; DOI:
10.1021/jm00319a005
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Totally Synthetic Steroid Hormones. V.1 (±)-2,3-Dimethoxyestra-1,3,5(10)-trien-17β-ol and Some Congeners
G. H. Douglas, C. R. Walk, and Herchel Smith
pp 27 - 29; DOI:
10.1021/jm00319a006
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Derivatives of Imidazole. II. Synthesis and Reactions of Imidazo[1,2-α]pyrimidines and Other Bi- and Tricyclic Imidazo Derivatives with Analgesic, Antiinflammatory, Antipyretic, and Anticonvulsant Activity
Luigi Almirante, Luigi Polo, Alfonso [ILL], Ercolina Provinciali, Pierluigi Rugarli, Afro Gamba, Amanda Olivi, and Walter Murmann
pp 29 - 33; DOI:
10.1021/jm00319a007
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Imidazoles. II. 5(or 4)-(Monosubstituted Triazeno)imidazole-4(or 5)-carboxamides
Y. Fulmer Shealy and Charles A. Krauth
pp 34 - 38; DOI:
10.1021/jm00319a008
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Synthesis and Pharmacological Properties of 1-Substituted 3-Dimethylaminoalkoxy-1H-indazoles
G. Palazzo, G. Corsi, L. Baiocchi, and B. Silvestrini
pp 38 - 41; DOI:
10.1021/jm00319a009
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Substituted s-Triazoles and Related Compounds
Harry L. Yale and Joseph J. Piala
pp 42 - 46; DOI:
10.1021/jm00319a010
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Iodinated 5- and 8-Hydroxyisoquinolines as Potential Amebicides
F. Schenker, R. A. Schmidt, W. Leimgruber, and A. Brossi
pp 46 - 48; DOI:
10.1021/jm00319a011
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4-Substituted Piperidines. III. Reduction of 1-Benzyl-4-cyano-4-t-aminopiperidines with Lithium Aluminium Hydride
Bert Hermans, Paul Van Daele, Cornelis van de Westeringh, Cyriel Van der Eycken, Jozef Boey, and Paul A. J. Janssen
pp 49 - 52; DOI:
10.1021/jm00319a012
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(-)-5-Ethyl-5-phenyl-2-pyrrolidinone. Unusual Reactions of 4-Nitro-4-phenylhexanoic Acid
P. M. G. Bavin
pp 52 - 55; DOI:
10.1021/jm00319a013
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9-Deamidooxytocin, an Analog of the Hormone Containing a Glycine Residue in Place of the Glycinamide Residue
Barbara M. Ferrier and Vincent du Vigneaud
pp 55 - 57; DOI:
10.1021/jm00319a014
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Synthesis of β-(4-Hydroxy-1-naphthyl)-DL-alanine
K. C. Tsou, Helen C. F. Su, R. B. Turner, and Ugo Mirachi
pp 57 - 60; DOI:
10.1021/jm00319a015
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β-(N-Piperazino)dimethylacetanilides and Their Local Anesthetic Activity
William O. Foye, Herbert B. Levine, and Walter L. McKenzie
pp 61 - 63; DOI:
10.1021/jm00319a016
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2-Hydroxyacetophenetidine, a New Metabolite of Acetophenetidine
A. Klutch, M. Harfenist, and A. H. Conney
pp 63 - 66; DOI:
10.1021/jm00319a017
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Nonclassical Antimetabolites. XXV.1 Inhibitors of Thymidine Kinase. I. A New Spectrophotometric Assay. Inhibition by Nucleoside Derivatives
B. R. Baker, Thomas J. Schwan, and Daniel V. Santi
pp 66 - 72; DOI:
10.1021/jm00319a018
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Nonclassical Antimetabolites. XXVI. Inhibitors of Thymidine Kinase. II.1,2 Inhibition by Functionalized 1-Alkyluracils
B. R. Baker and Thomas J. Schwan
pp 73 - 76; DOI:
10.1021/jm00319a019
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Carcinogenicity of Epoxides, Lactones, and Peroxy Compounds. III. Biological Activity and Chemical Reactivity
B. L. Van Duuren and B. M. Goldschmidt
pp 77 - 79; DOI:
10.1021/jm00319a020
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Synthesis and Study of β-Chloroethylamines, Sulfides, and Sulfones Structurally Related to Dibenzyline
Samuel Lamdan, Carlos M. Vega, and Carlos H. Gaozza
pp 79 - 83; DOI:
10.1021/jm00319a021
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Synthesis of Potentially Cytoactive Amino Acid Amide Mustards
Harold Z. Sommer, Charles Scher, Shlomo Bien, Gert Olsen, Jiban K. Chakrabarti, and Orrie M. Friedman
pp 84 - 88; DOI:
10.1021/jm00319a022
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Sulfonanilides. I. Monoalkyl- and Arylsulfonamidophenethanolamines
Robert H. Uloth, Jerry R. Kirk, William A. Gould, and A. A. Larsen
pp 88 - 97; DOI:
10.1021/jm00319a023
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Synthesis and Properties of 5-Mercaptomethyluracil and Related Derivatives
Alfredo Giner-Sorolla and Lillian Medrek
pp 97 - 101; DOI:
10.1021/jm00319a024
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Nucleosides. XXIX. 1-β-D-Arabinofuranosyl-5-fluorocytosine and Related Arabino Nucleosides
Jack J. Fox, Naishun Miller, and Iris Wempen
pp 101 - 105; DOI:
10.1021/jm00319a025
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3-Deaza-6-methylthiopurine Ribonucleoside
John A. Montgomery and Kathleen Hewson
pp 105 - 107; DOI:
10.1021/jm00319a026
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5-Arylaminopyrimidines
Fred R. Gerns, Agostino Perrotta, and George H. Hitchings
pp 108 - 115; DOI:
10.1021/jm00319a027
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Pyridine Chemistry. II. Further Studies on the Smiles Rearrangement of the 3-Amino-2,2′-dipyridyl Sulfide System. The Synthesis of Some 1,6-Diazaphenothiazines
Oscar R. Rodig, Richard E. Collier, and Robert K. Schlatzer
pp 116 - 120; DOI:
10.1021/jm00319a028
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Pyrimidines. XVI. 2,4,5-Triaminopyrimidines and Related Compounds
Darrell E. O'Brien, C. Wayne Noell, Roland K. Robins, and C. C. Cheng
pp 121 - 126; DOI:
10.1021/jm00319a029
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4-(2-Piperidyl)-1,3-dioxolanes with Local Anesthetic, Spasmolytic, and Central Nervous System Activity
W. R. Hardie, J. Hidalgo, I. F. Halverstadt, and R. E. Allen
pp 127 - 136; DOI:
10.1021/jm00319a030
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3-Indolylsuccinimides and 3-(3-Pyrrolidinyl)indoles
Y. G. Perron, W. F. Minor, M. E. Bierwagen, S. A. Ridlon, and M. H. Pindell
pp 136 - 140; DOI:
10.1021/jm00319a031
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DL-2-Amino-4-(4-pyridyl)butyric Acid
Frederick Leonard and Walter Tschannen
pp 140 - 140; DOI:
10.1021/jm00319a032
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5-Nitro- and 5-Aminogramines
Joseph I. DeGraw, Vernon H. Brown, and W. A. Skinner
pp 140 - 142; DOI:
10.1021/jm00319a033
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Substitution in the Hydantoin Ring. III. Bicyclo[3.3.0]octane Derivatives
Meldrum B. Winstead, Frederick R. Scholer, and Kenneth H. Wildrick
pp 142 - 143; DOI:
10.1021/jm00319a034
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Synthesis and Biological Activity of 9-β-D-Ribofuranosyl-6-hydroxylaminopurine
Alfredo Giner-Sorolla, Lillian Medrek, and Aaron Bendich
pp 143 - 144; DOI:
10.1021/jm00319a035
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N-Substituted Ureidobis(1-aziridinyl)phosphine Oxides
Rudi Rätz and Miriam Gruber
pp 144 - 146; DOI:
10.1021/jm00319a036
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9,10-Seco-10-methylestrone
S. Mahapatra and R. M. Dodson
pp 147 - 149; DOI:
10.1021/jm00319a037
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Synthesis of Some Homologs of Fluoropyruvic Acid and Their Effect on the Carbohydrate Metabolism of Ehrlich Ascites Tumor and on Lactate Dehydrogenase
D. R. Grassetti, M. E. Brokke, and J. F. Murray
pp 149 - 151; DOI:
10.1021/jm00319a038
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Preparation of Some ω-(Pyridylalkyl)benzamide and Benzoate Derivatives
O. H. Hankovszky and K. Hideg
pp 151 - 153; DOI:
10.1021/jm00319a039
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Synthesis of 1,4-Disubstituted Piperazines. I
Matthew Verderame
pp 153 - 154; DOI:
10.1021/jm00319a040
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Synthesis and Antifertility Activity of 5-(Phenoxymethyl)-2-oxazolidinethiones
Gilbert A. Youngdale, Gordon W. Duncan, D. Edward Emmert, and Daniel Lednicer
pp 155 - 157; DOI:
10.1021/jm00319a041
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The Osmium Tetroxide Catalyzed Hydroxylation of 1,4-Dimethylenecyclohexanes
James G. Murphy
pp 157 - 159; DOI:
10.1021/jm00319a042
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Synthesis of β-5-Fluoro-2′-deoxyuridylyl-(5′→5′)-β-5-fluoro-2′- deoxyuridine
David G. Parsons and Charles Heidelberger
pp 159 - 159; DOI:
10.1021/jm00319a043
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The Synthesis of Some 8-Alkylthio-2-thiotheophyllines and 8-Alkylthio-6-thiotheophyllines
Albert J. Dietz and Raymond M. Burgison
pp 160 - 160; DOI:
10.1021/jm00319a044
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Benzo[a][3,6]phenanthrolines
Robert T. Parfitt
pp 161 - 162; DOI:
10.1021/jm00319a045
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Cyclohexylammonium Hydrogen N-2-Chloroethyl-N-5-chloro(1-chloromethyl)pentyl Phosphorodiamidate
Gert Olsen and Orrie M. Friedman
pp 162 - 162; DOI:
10.1021/jm00319a046
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Synthesis of the Di-N-phenyl- and Di-N-(α-naphthyl)urethans of 1,1-Dimethylol-3-cyclopentene
Edward J. Grubbs
pp 162 - 163; DOI:
10.1021/jm00319a047
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Syntheses of 3-Cyano-3-methyl-4-thiochromanone and 3-Carbomethoxy-3-methyl-4-thiochromanone
Tosio Moriwake
pp 163 - 164; DOI:
10.1021/jm00319a048
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The Partial Synthesis of 1,2,3,4,4aα,9,10,10aβ-Octahydro-1α-(2-hydroxyethyl)-7-methoxy-2β- methyl-2α-phenanthrenecarboxylic Acid δ-Lactone
Joseph C. Touchstone, John R. Grunwell, William H. Elliott, and Sidney A. Thayer
pp 164 - 165; DOI:
10.1021/jm00319a049
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Myelographic Agents. II. Some Iodophthalates
J. H. Ackerman, V. Akullian, C. Moore, and A. A. Larsen
pp 165 - 168; DOI:
10.1021/jm00319a050
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A. Readings in Pharmacology. B. Pharmacy in History.
Alfred Burger
pp 168 - 168; DOI:
10.1021/jm00319a051
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Advances in Pharmacology. Volume 3.
Alfred Bu
pp 168 - 168; DOI:
10.1021/jm00319a052
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Issue 2


Synthesis and Pharmacological Properties of 9-Decarboxamido-oxytocin
Luis A. Branda and Vincent du Vigneaud
pp 169 - 172; DOI:
10.1021/jm00320a001
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Mammalian Antifertility Agents. III. 1-Aryl-2-phenyl-1,2,3,4-tetrahydro-1-naphthols, 1-Aryl-2-phenyl-3,4-dihydronaphthalenes, and Their Derivatives
Daniel Lednicer, Stanley C. Lyster, Brooke D. Aspergren, and Gordon W. Duncan
pp 172 - 176; DOI:
10.1021/jm00320a002
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α,β-Diphenyl-α-trifluoromethyl-2-pyridineethanol and Related Compounds as Synthetic Estrogens
John R. Dice, Lorraine Scheinman, and Kay W. Berrodin
pp 176 - 178; DOI:
10.1021/jm00320a003
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Ring-D-Bridged Steroid Analogs. II.1 14α,17α-Etheno-16α-carbomethoxypregn-4-ene-3,20-dione2
A. J. Solo and Baldev Singh
pp 179 - 181; DOI:
10.1021/jm00320a004
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Derivatives of Piperazine. XXXV.1a Synthesis of 2-Phenylpiperazine and Some Derivatives
William R. Roderick, Howard J. Platte, and C. B. Pollard
pp 181 - 185; DOI:
10.1021/jm00320a005
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Derivatives of 2-Azabicyclo [2.2.2]octane. I
Frank J. Villani and Claire A. Ellis
pp 185 - 187; DOI:
10.1021/jm00320a006
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Analgetic Activity of Some δ-Amino Ketones And Their Derivatives
David L. Goldhamer, Anthony W. Pircio, Armin Wilson, and Leonard Weintraub
pp 187 - 191; DOI:
10.1021/jm00320a007
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Substituted 2,3-Dihydro-1,5-benzothiazepin-4(5H)-one and Related Compounds. II. A New Class of Antidepressants
John Krapcho and Chester F. Turk
pp 191 - 195; DOI:
10.1021/jm00320a008
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Aziridine Derivatives as Potential Monoamine Oxidase Inhibitors
J. N. Wells, A. V. Shirodkar, and A. M. Knevel
pp 195 - 197; DOI:
10.1021/jm00320a009
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Synthesis of Chelating Compounds to Be Used as Potential Bone Seekers
Gad Shtacher and William Taub
pp 197 - 203; DOI:
10.1021/jm00320a010
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Quantification and Prediction of the Biological Activities of Chloramphenicol Analogs by Microbial Kinetics
Edward R. Garrett, Olga K. Wright, George H. Miller, and Kenneth L. Smith
pp 203 - 208; DOI:
10.1021/jm00320a011
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Antibacterial Activity of Compounds with Both Mercury and Tin in Organic Combination
V. L. Miller and A. C. Jerstad
pp 208 - 210; DOI:
10.1021/jm00320a012
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Antiviral Agents. II. Substituted Morpholinium Quaternary Salts
Elvin L. Anderson, John E. Casey, Elizabeth E. Force, Erling M. Jensen, Ralph S. Matz, and Donald E. Rivard
pp 211 - 213; DOI:
10.1021/jm00320a013
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Dipeptide Nitrogen Mustards of Glycine and γ-Aminobutyric Acid
S.-C. J. Fu, H. Terzian, C. L. Maddock, and V. M. Binns
pp 214 - 216; DOI:
10.1021/jm00320a014
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Heterocyclic Derivatives of 2-Chloroethyl Sulfide with Antitumor Activity
Richard M. Peck, Anna P. O'Connell, and Hugh J. Creech
pp 217 - 221; DOI:
10.1021/jm00320a015
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Synthesis, Chemistry, and Preliminary Pharmacology of Arsenical Nitrogen Mustards and Structurally Related Nonalkylating Arsenicals
Thomas J. Bardos, Nirmalendu Datta-Gupta, and Peter Hebborn
pp 221 - 227; DOI:
10.1021/jm00320a016
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Synthesis and Carcinolytic Activity of Some Diaryliodonium Salts
Robert A. Wiley and Maureen A. Salter
pp 228 - 231; DOI:
10.1021/jm00320a017
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Synthesis of Potential Antineoplastic Agents. XXXV. Phosphorus-Containing Structural Analogs of Myleran
Robert F. Struck
pp 231 - 234; DOI:
10.1021/jm00320a018
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Nucleosides from Homoribose
John A. Montgomery and Kathleen Hewson
pp 234 - 237; DOI:
10.1021/jm00320a019
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Preparation and Antitumor Activity of Olivacine and Some New Analogs
Carol W. Mosher, Osborne P. Crews, Edward M. Acton, and Leon Goodman
pp 237 - 241; DOI:
10.1021/jm00320a020
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Compounds Derived from L-Threitol 1,4-Bismethanesulfonate
Peter W. Feit
pp 241 - 242; DOI:
10.1021/jm00320a021
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Synthesis of Grisan and Coumaran-3-one Derivatives with Potential Insect-Repellent Properties
Vasu Dev, Ronald P. Quintana, and Andrew Lasslo
pp 242 - 244; DOI:
10.1021/jm00320a022
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The Synthesis of p-Guanidinobenzamidines
Victor J. Bauer and S. R. Safir
pp 244 - 246; DOI:
10.1021/jm00320a023
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The Chemical Structure of a Cocarcinogen and of Phorbol Isolated from Croton Oil
E. Hecker, H. Kubinyi, H. Bresch, and Ch. von Szczepanski
pp 246 - 247; DOI:
10.1021/jm00320a024
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Biologically Active Guanidines and Related Compounds. III.1 Some Aryloxyalkylurea Derivatives
G. J. Durant and S. H. B. Wright
pp 247 - 248; DOI:
10.1021/jm00320a025
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The Synthesis and Pharmacological Activity of 5-Ethyl-5-(3-hydroxy-1-methylbutyl)barbituric Acid
Y. J. Dickert, P. J. Shea, and L. P. McCarty
pp 249 - 249; DOI:
10.1021/jm00320a026
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The Synthesis of 3-Fluoroestra-1,3,5(10)-trienes
Duane F. Morrow and Ruthann M. Hofer
pp 249 - 251; DOI:
10.1021/jm00320a027
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Synthesis of Some Substituted Tryptophols of Possible Physiological Importance and a Study with 3-(2-Acetoxyethyl)-5-methoxyindole (5-Methoxytryptophol O-Acetate) on Sexual Maturation
Robert G. Taborsky and Peter Delvigs
pp 251 - 254; DOI:
10.1021/jm00320a028
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Heterocyclic Amines. III. 3-Dimethylaminofuran
John D. Prugh and Walter C. McCarthy
pp 254 - 255; DOI:
10.1021/jm00320a029
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Poly-L-α,γ-diaminobutyric Acid Hydrochloride
Margaret J. Fridecky and William H. McGregor
pp 255 - 256; DOI:
10.1021/jm00320a030
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Sulfamylsemicarbazide Hypoglycemic Agents. IV
J. M. McManus and C. F. Gerber
pp 256 - 257; DOI:
10.1021/jm00320a031
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Synthetic Biologically Active Polymers. III. A Sulfapyridine-Formaldehyde Copolymer
L. Guy Donaruma and John Razzano
pp 258 - 259; DOI:
10.1021/jm00320a032
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Synthesis of Substituted β-Lactams
B. G. Chatterjee and P. N. Moza
pp 259 - 261; DOI:
10.1021/jm00320a033
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The Role of Analgesic Drug Metabolites in the Formation of Lens Opacities
Vernon H. Brown, Joseph I. DeGraw, Samuel A. Ferguson, and W. A. Skinner
pp 261 - 261; DOI:
10.1021/jm00320a034
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The Synthesis of Tritium-Labeled Phenoxybenzamine Hydrochloride
Jon E. Lewis and Jack W. Miller
pp 261 - 262; DOI:
10.1021/jm00320a035
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Silicon-Substituted Medicinal Agents. Phenyl-Substituted Silacarbamates
Ralph J. Fessenden and Marvin D. Coon
pp 262 - 263; DOI:
10.1021/jm00320a036
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Isomeric Estranes
R. E. Counsell
pp 263 - 263; DOI:
10.1021/jm00320a037
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Synthesis of Arysulfonyl-1-methyl-S-isothiosemicarbazides
Carlos Sunkel and Sonia Erazo
pp 263 - 264; DOI:
10.1021/jm00320a038
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A New Naphthylacetamide Derivative
Tiberio Bruzzese and Carla Turba
pp 264 - 264; DOI:
10.1021/jm00320a039
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Derivatives of 2-Azabicyclo[2.2.2]octane. II
Frank J. Villani and Claire A. Ellis
pp 264 - 265; DOI:
10.1021/jm00320a040
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Substitution in the Hydantoin Ring. IV. N-3-p-Bromoanilinomethyl Derivatives
Meldrum B. Winstead
pp 265 - 266; DOI:
10.1021/jm00320a041
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Quinoxaline Studies. XIII. N-(2-Quinoxaloyl)-α-amino Acids
Shlomo Gerchakov, Peter J. Whitman, and Harry P. Schultz
pp 266 - 268; DOI:
10.1021/jm00320a042
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The Acetylation of 1-(β-D-Arabinofuranosyl)cytosine
Abelardo P. Martinez, William W. Lee, and Leon Goodman
pp 268 - 268; DOI:
10.1021/jm00320a043
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Potential Antifibrillatory Agents. N-(ω-Aminoalkoxy)phthalimides
Milton J. Kornet
pp 269 - 269; DOI:
10.1021/jm00320a044
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Progress in Drug Research. Volume 8.
Alfred Burger
pp 270 - 270; DOI:
10.1021/jm00320a045
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Selective Toxicity.
Alfred Burger
pp 270 - 270; DOI:
10.1021/jm00320a046
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Cyclophosphamide (Cytoxan).
Frank D. Popp
pp 270 - 270; DOI:
10.1021/jm00320a047
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New Drugs.
Alfred Burger
pp 270 - 270; DOI:
10.1021/jm00320a048
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Issue 3


The Chemorelease of Norepinephrine from Mouse Hearts. Structure-Activity Relationships. I. Sympathomimetic and Related Amines
J. W. Daly, C. R. Creveling, and B. Witkop
pp 273 - 280; DOI:
10.1021/jm00321a001
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The Chemorelease of Norepinephrine in Mouse Hearts. Structure-Activity Relationships. II. Drugs Affecting the Sympathetic and Central Nervous Systems
J. W. Daly, C. R. Creveling, and B. Witkop
pp 280 - 284; DOI:
10.1021/jm00321a002
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The Depletion of Norepinephrine-3H from Heart by α-Methyl-m-tyrosine. A Novel and Convenient Method for Assaying the Inhibition of Aromatic Amino Acid Decarboxylase in Vivo
C. R. Creveling, J. W. Daly, and B. Witkop
pp 284 - 286; DOI:
10.1021/jm00321a003
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Metabolism of Metaxalone
Robert B. Bruce, Lennox Turnbull, Jack Newman, and Jefferson Pitts
pp 286 - 288; DOI:
10.1021/jm00321a004
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Design and Synthesis of Thiolesters for the Histochemical Demonstration of Esterase and Lipase via the Formation of Osmiophilic Diazo Thioethers
Jacob S. Hanker, Lionel Katzoff, Howard R. Rosen, Myron L. Seligman, Hiromi Ueno, and Arnold M. Seligman
pp 288 - 291; DOI:
10.1021/jm00321a005
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Histamine Releasers. I. Structure of the Dimer Formed from p-Methoxy-N-methylphenethylamine and Formaldehyde
Joseph I. DeGraw, Vernon H. Brown, Samuel A. Ferguson, Nicholas E. Kontaxis, and W. A. Skinner
pp 292 - 294; DOI:
10.1021/jm00321a006
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Electronic Structures of Some N-Alkyl-Substituted Amides of Interest as Cholinesterase Inhibitors
William Paul Purcell
pp 294 - 297; DOI:
10.1021/jm00321a007
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Application of Partition Coefficients, Electric Moments, Electronic Structures, and Free-Energy Relationships to the Interpretation of Cholinesterase Inhibition
William P. Purcell, James G. Beasley, Ronald P. Quintana, and Judith A. Singer
pp 297 - 303; DOI:
10.1021/jm00321a008
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Octahydrophenanthrene Analogs of Tetrabenazine
K. E. Fahrenholtz, A. Capomaggi, M. Lurie, M. W. Goldberg, and R. W. Kierstead
pp 304 - 310; DOI:
10.1021/jm00321a009
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The Syntheses and Hypotensive Activities of Some Substituted 1,4-Diazabicyclo[4.4.0]decanes
Alan D. Lourie and Allan R. Day
pp 311 - 315; DOI:
10.1021/jm00321a010
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Synthesis and Antiinflammatory Activity of a Series 1-Aryl-2-pyrrolidinone Derivatives
K. Okumura, I. Inoue, M. Ikezaki, G. Hayashi, S. Nurimoto, and K. Shintomi
pp 315 - 319; DOI:
10.1021/jm00321a011
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Synthesis of trans-2-Cyclohexyloxycyclopropylamine and Derivatives
Jacob Finkelstein, Elliot Chiang, F. M. Vane, and John Lee
pp 319 - 323; DOI:
10.1021/jm00321a012
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Hypocholesterolemic Agents. VI.1 A- and B-Ring-Modified Azacholesterols
P. D. Klimstra, R. E. Ranney, and R. E. Counsell
pp 323 - 326; DOI:
10.1021/jm00321a013
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The Synthesis of Potential Anabolic Agents. Steroidal Oxadiazoles
Robert E. Havranek, G. Brooke Hoey, and David H. Baeder
pp 326 - 328; DOI:
10.1021/jm00321a014
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The Relationship between Structure and Activity in a Novel Series of Serum Cholesterol-Lowering Agents
L. G. Humber, C. I. Chappel, A. V. Marton, M. Kraml, and J. Dubuc
pp 329 - 337; DOI:
10.1021/jm00321a015
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Totally Synthetic Steroid Hormones. VII.1 Some (±)-8α-Estrane and (±)-13β-Alkyl-8α-gonane Derivatives
G. C. Buzby, E. Capaldi, G. H. Douglas, D. Hartley, D. Herbst, G. A. Hughes, K. Ledig, J. McMenamin, T. Pattison, Herchel Smith, C. R. Walk, and G. R. Wendt
pp 338 - 341; DOI:
10.1021/jm00321a016
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Synthesis and Pharmacological Activity of Alkylated Tryptamines
Asher Kalir and Stephen Szara
pp 341 - 344; DOI:
10.1021/jm00321a017
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Synthesis and Biological Activity of Some 5-, 6-, and 7-Aminomethyl-2,3-dimethylindoles
R. W. Brimblecombe, D. F. Downing, and R. R. Hunt
pp 345 - 347; DOI:
10.1021/jm00321a018
PDF
Hexahydropyrimidines. VII.1 A Study of 2-Substituted 1,3-Bis(2-hydroxy-3-methoxybenzyl)hexahydropyrimidines and 2-Substituted 1,3-Bis(3,4-dimethoxybenzyl)hexahydropyrimidines as Antitumor Agents2
John H. Billman and M. Sami Khan
pp 347 - 351; DOI:
10.1021/jm00321a019
PDF
3-Substituted 2-Thiohydrouracils. Synthesis and Antitubercular and Antineoplastic Activities
Arthur C. Glasser and Richard M. Doughty
pp 351 - 353; DOI:
10.1021/jm00321a020
PDF
1-Deaza-6-methylthiopurine Ribonucleoside
John A. Montgomery and Kathleen Hewson
pp 354 - 357; DOI:
10.1021/jm00321a021
PDF
Potential Carcinolytic Agents.1 III. Fluoronitrogen Mustard Analogs of Cyclophosphamide2
Zinon B. Papanastassiou, Robert J. Bruni, Frances Potts Fernandes, and Philip L. Levins
pp 357 - 359; DOI:
10.1021/jm00321a022
PDF
Phosphorus Mustards. II. The Synthesis and Biological Evaluation of Bis(2-chloroethyl)methylphosphine Hydrochloride
D. C. Smith, A. H. Soloway, and R. W. Turner
pp 360 - 362; DOI:
10.1021/jm00321a023
PDF
Attempted Synthesis of 2,4-Dihydroxy-4,3-borazaropyridine. Preparation of Aminoalkylboronic Acids
D. N. Butler and A. H. Soloway
pp 362 - 365; DOI:
10.1021/jm00321a024
PDF
Nucleosides. III. Studies on 5-Methylamino-2′-deoxyuridine as a Specific Antiherpes Agent
T. Y. Shen, J. F. McPherson, and B. O. Linn
pp 366 - 369; DOI:
10.1021/jm00321a025
PDF
Anticancer and Potential Antiviral Activity of Complex Inorganic Compounds
Stanley Kirschner, Yung-Kang Wei, Dawn Francis, and John G. Bergman
pp 369 - 372; DOI:
10.1021/jm00321a026
PDF
Purine Sulfonamides
Alden G. Beaman, William Tautz, Robert Duschinsky, and E. Grunberg
pp 373 - 378; DOI:
10.1021/jm00321a027
PDF
Synthetic Schistosomicides. VIII. N-Mono- and N,N-Dialkyl-N′-(4-arylazo-1-naphthyl)alkylenediamines and Related Compounds
Edward F. Elslager, David B. Capps, Dianne H. Kurtz, Franklin W. Short, Leslie M. Werbel, and Donald F. Worth
pp 378 - 391; DOI:
10.1021/jm00321a028
PDF
Reactions of Mercaptoamines. III. Synthesis of N-Monosubstituted 2-Mercaptoethylamines
Arthur F. Ferris, O. LeRoy Salerni, and Beverly A. Schutz
pp 391 - 394; DOI:
10.1021/jm00321a029
PDF
Radioprotective Activity of Triammonium 2-Dithiocarbamoyl-3-dithiocarbonylthiopropanoate
Richard I. H. Wang, William Dooley, William O. Foye, and James Mickles
pp 394 - 396; DOI:
10.1021/jm00321a030
PDF
Organic Disulfides and Related Substances. XVII.1a Analogs of o-(2-Aminoethyldithio)benzoic Acid as Antiradiation Drugs1b
Lamar Field and H. K. Kim
pp 397 - 402; DOI:
10.1021/jm00321a031
PDF
5,6-Dihydro-3-(5-nitro-2-furyl)imidazo[2,1-b]thiazoles and Acid Addition Salts
Harry R. Snyder and Louis E. Benjamin
pp 402 - 405; DOI:
10.1021/jm00321a032
PDF
Nitrofuryl Heterocycles. III.1 3-Alkyl-5-(5-nitro-2-furyl)-1,2,4-triazoles and Intermediates
Homer A. Burch and Warren O. Smith
pp 405 - 408; DOI:
10.1021/jm00321a033
PDF
Nitrofuryl Heterocycles. IV1. 4-Amino-2-(5-nitro-2-furyl)quinazoline Derivatives
Homer A. Burch
pp 408 - 410; DOI:
10.1021/jm00321a034
PDF
Carboranes. I. Nitrogen Mustards
A. H. Soloway and D. N. Butler
pp 411 - 412; DOI:
10.1021/jm00321a035
PDF
L-(+)-2β-Tropanyl Diphenylborinate
Edward R. Atkinson, Donna L. Mc Ritchie, and A. H. Soloway
pp 412 - 414; DOI:
10.1021/jm00321a036
PDF
Tertiary Phosphines and Phosphine Oxides Containing a 2-Haloethyl Group
Robert F. Struck and Y. Fulmer Shealy
pp 414 - 416; DOI:
10.1021/jm00321a037
PDF
Glycerol 1,3- and 1,2,4-Butanetriol 1,4-Bismethanesulfonates
Peter W. Feit and Ole Tvaermose Nielsen
pp 416 - 417; DOI:
10.1021/jm00321a038
PDF
v-Triazolo[4,5-d]pyrimidines. III. N-(3-Alkyl-5-amino-3H-v-triazolo[4,5-d]pyrimidin-7-yl)-amino Acids
Y. Fulmer Shealy, C. Allen O'Dell, and John A. Montgomery
pp 417 - 419; DOI:
10.1021/jm00321a039
PDF
6-Azauracil Derivatives of Fluoropyruvic Acid
G. J. Durr
pp 419 - 420; DOI:
10.1021/jm00321a040
PDF
The Synthesis and Antitumor Activity of Several Thiosemicarbazones Related to Kethoxal Bis(thiosemicarbazone)
H. G. Petering, G. J. VanGiessen, J. A. Crim, and H. H. Buskirk
pp 420 - 421; DOI:
10.1021/jm00321a041
PDF
Synthesis of Potential Antineoplastic Agents. XIII. 1-{p-[Bis(2-chloroethyl)amino]benzyl}-pyridinium p-Toluenesulfonate and Related Compounds
Dru W. Alwani, Adria Catala Noble, and Frank D. Popp
pp 421 - 423; DOI:
10.1021/jm00321a042
PDF
2,4-Bis(arylamino)pyrimidines as Antimicrobial Agents
Dolly Ghosh
pp 423 - 424; DOI:
10.1021/jm00321a043
PDF
Nitrofuryl Heterocycles. II.1 2-Alkyl-6-(5-nitro-2-furyl)-3(2H)-pyridazinones and 4,5-Dihydro Derivatives
Homer A. Burch and Louis E. Benjamin
pp 425 - 426; DOI:
10.1021/jm00321a044
PDF
The Bacteriostatic Effectiveness of 1-Alkyl-3-(3,4-dichlorophenyl)ureas
Thomas A. Schenach, James Brown, Allen J. Wysocki, and Frank Yackovich
pp 426 - 428; DOI:
10.1021/jm00321a045
PDF
Halonitroanilides and Their Bacteriostatic Activity
Joseph W. Baker, Ignatius Schumacher, Gerald L. Bachman, Daniel P. Roman, and Alan L. Tharp
pp 428 - 430; DOI:
10.1021/jm00321a046
PDF
Derivatives of 5-Carboxymethylthiazolidine-2,4-dione, a New Group of Antiviral Compounds
A. Krbavčič, M. Plut, A. Pollak, M. Tišler, M. Likar, and P. Schauer
pp 430 - 431; DOI:
10.1021/jm00321a047
PDF
3-Aryl-5-halomethylisoxazoles. A New Class of Anthelmintics
H. G. Sen, D. Seth, U. N. Joshi, and P. Rajagopalan
pp 431 - 433; DOI:
10.1021/jm00321a048
PDF
Syntheses and Properties of Mono-, Di-, and Tritestosteroxysilanes
Edward Chang and Vijay K. Jain
pp 433 - 435; DOI:
10.1021/jm00321a049
PDF
Some Alkylideneaminooxyalkanoic Acids and Derivatives
L. H. Klemm and D. Hsu Lee
pp 435 - 436; DOI:
10.1021/jm00321a050
PDF
Compounds Affecting the Central Nervous System. II. Substituted 1,2,3,4-Tetrahydropyrido[4,3-b]indoles
R. G. W. Spickett
pp 436 - 438; DOI:
10.1021/jm00321a051
PDF
Indole Hydrazides as Potential Monoamine Oxidase Inhibitors
T. Nogrady and L. Morris
pp 438 - 439; DOI:
10.1021/jm00321a052
PDF
DL-2-Hydrazino-3-(4-hydroxyphenyl)propionic Acid
Joseph D. Benigni and Donald E. Dickson
pp 439 - 440; DOI:
10.1021/jm00321a053
PDF
2-Methyl-3-phenoxycyclopropylamine
Jacob Finkelstein, Elliot Chiang, and John Lee
pp 440 - 441; DOI:
10.1021/jm00321a054
PDF
Agents Affecting Lipid Metabolism. XXI. Miscellaneous Compounds Related to trans-1,4-Bis(2-chlorobenzylaminomethyl)cyclohexane
Leslie G. Humber
pp 441 - 443; DOI:
10.1021/jm00321a055
PDF
t-Butyl Ester of 7-Aminocephalosporanic Acid
R. John Stedman
pp 444 - 444; DOI:
10.1021/jm00321a056
PDF
Some Ureas and Urethans Derived from p-Aminophenol
Carol W. Mosher, Edward M. Acton, and Leon Goodman
pp 444 - 445; DOI:
10.1021/jm00321a057
PDF
The Six Trimethoxyphenylisopropylamines (Trimethoxyamphetamines)
Alexander T. Shulgin
pp 445 - 446; DOI:
10.1021/jm00321a058
PDF
Substrates for Cytochemical Demonstration of Enzyme Activity. II. Some Dihalo-3-indolyl Phosphates and Sulfates
Jerome P. Horwitz, Jonathan Chua, Michael Noel, Joseph T. Donatti, and Josef Freisler
pp 447 - 447; DOI:
10.1021/jm00321a059
PDF
N-Substituted DL-Aspartic Acids and β-Methyl Esters
Marvin J. Karten, Ernest Magnien, Allan Schwinn, and Seymour L. Shapiro
pp 447 - 448; DOI:
10.1021/jm00321a060
PDF
N-[(4-Tolysulfonyl)carbamoyl]amino Acids
Marvin J. Karten, Allan Schwinn, and William Oroshnik
pp 448 - 449; DOI:
10.1021/jm00321a061
PDF
Substituted 2-Phenoxypropionic and -butyric Acids and Derivatives
E. Magnien, F. Testa, and S. L. Shapiro
pp 449 - 450; DOI:
10.1021/jm00321a062
PDF
The Chemistry of Natural Products. Volume VI, The Chemistry of the Vitamins.
Arthur F. Wagner
pp 451 - 451; DOI:
10.1021/jm00321a063
PDF
Animals Parasitic in Man.
J. Allan Waitz
pp 451 - 451; DOI:
10.1021/jm00321a064
PDF
International Series of Monographs on Child Psychiatry. Volume III. Drug Addiction in Youth.
Everette L. May
pp 451 - 452; DOI:
10.1021/jm00321a065
PDF
The United States Pharmacopeia.
Warren E. Weaver
pp 452 - 452; DOI:
10.1021/jm00321a066
PDF
Evaluation of Drug Activities: Pharmacometrics.
Alfred Burger
pp 452 - 452; DOI:
10.1021/jm00321a067
PDF
Progress in Medicinal Chemistry. Volume 4.
Alfred Burger
pp 452 - 452; DOI:
10.1021/jm00321a068
PDF

Issue 4


Stereochemical Aspects of Analgetics. Preparation of Isomeric 1-Methyl-4-phenyl-trans-decahydro-4-propionoxyquinolines
Edward E. Smissman and Martin Steinman
pp 455 - 457; DOI:
10.1021/jm00322a001
PDF
Conformational Aspects of Acetylcholine Receptor Sites. The Isomeric 3-Trimethylammonium-2-acetoxy-trans-decalin Halides1 and the Isomeric α,β-Dimethylacetylcholine Halides2
Edward E. Smissman, Wendel L. Nelson, Jules B. LaPidus, and James L. Day
pp 458 - 465; DOI:
10.1021/jm00322a002
PDF
Comparison of the Hypotensive Activities of Highly Hindered Open-Chain Amines and Their Cyclic Counterparts
Nelson R. Easton, Francis G. Henderson, Walter J. McMurray, and Nelson J. Leonard
pp 465 - 468; DOI:
10.1021/jm00322a003
PDF
1-Ethynylphenethylamine
Alfred Burger, Stuart E. Zimmerman, and E. J. Ariëns
pp 469 - 470; DOI:
10.1021/jm00322a004
PDF
The Influence of Some 1-Substituted 6-Methoxy-1,2,3,4-tetrahydro-β-carbolines on the Metabolism and Activity of 5-Hydroxytryptamine
Ryszard J. Gryglewski, Stanislaw H. Misztal, Jacek A. Splawiński, and Bogumila Panczenko
pp 471 - 474; DOI:
10.1021/jm00322a005
PDF
2H-1,4-Benzoxazin-2-ones
Robert Bruce Moffett
pp 475 - 478; DOI:
10.1021/jm00322a006
PDF
2-Amino-5-Substituted 1,3,4-Oxadiazoles and 5-Imino-2-Substituted Δ2-1,3,4-Oxadiazolines. A Group of Novel Muscle Relaxants
Harry L. Yale and Kathryn Losee
pp 478 - 483; DOI:
10.1021/jm00322a007
PDF
Compounds Acting on the Central Nervous System. IV. 4-Substituted 2,3-Polymethylenequinolines
G. K. Patnaik and M. M. Vohra
pp 483 - 488; DOI:
10.1021/jm00322a008
PDF
Thietane 1,1-Dioxides
Jack N. Wells and Frank S. Abbott
pp 489 - 492; DOI:
10.1021/jm00322a009
PDF
New Local Anesthetics.1 I. Esters of 1,2-Diethyl-3-hydroxymethylpyrazolidine
Milton J. Kornet
pp 493 - 495; DOI:
10.1021/jm00322a010
PDF
Synthesis and Biological Activity of 7-Bromo-8-methyl-10-(1-D-ribityl)isoalloxazine, an Analog of Riboflavin
R. D. Faulkner and J. P. Lambooy
pp 495 - 497; DOI:
10.1021/jm00322a011
PDF
Synthesis and Pharmacological Activity of 4-D-Glutamine-oxytocin,1 5-D-Asparagine-oxytocin, and 4-D-Glutamine-5-D-asparagine-oxytocin
A. S. Dutta, Nitya Anand, and K. Kar
pp 497 - 499; DOI:
10.1021/jm00322a012
PDF
The Synthesis and Pharmacologic Evaluation of a Series of 8-Alkylthio-Thiated Theophyllines
Albert J. Dietz and Raymond M. Burgison
pp 500 - 506; DOI:
10.1021/jm00322a013
PDF
The Metabolic Fate of Tolbutamide in Man and in the Rat
Richard C. Thomas and George J. Ikeda
pp 507 - 510; DOI:
10.1021/jm00322a014
PDF
The Preparation and Chemistry of 9α,10α-Oxidoestra-4-en-3-ones
E. Farkas and J. M. Owen
pp 510 - 512; DOI:
10.1021/jm00322a015
PDF
Antiinflammatory Δ4-Pregnenolone Derivatives
R. Deghenghi, M. Boulerice, J. G. Rochefort, S. N. Sehgal, and D. J. Marshall
pp 513 - 516; DOI:
10.1021/jm00322a016
PDF
Derivatives of 3,4-Diphenylchromanes as Estrogens and Implantation Inhibitors
Richard W. J. Carney, William L. Bencze, Janice Wojtkunski, Alfred A. Renzi, Louis Dorfman, and George DeStevens
pp 516 - 520; DOI:
10.1021/jm00322a017
PDF
Effect of Organic Compounds on Reproductive Processes. III. Alkylating Agents Derived from Various Diamines
W. A. Skinner, M. Cory, T. E. Shellenberger, and J. I. DeGraw
pp 520 - 522; DOI:
10.1021/jm00322a018
PDF
Insect Chemosterilants. III. 1-Aziridinylphosphine Oxides
Alexej B. Bořkovec, Charles W. Woods, and Richard T. Brown
pp 522 - 526; DOI:
10.1021/jm00322a019
PDF
Synthesis and Antiinflammatory Activity of 2,3-Bis(p-methoxyphenyl)indole and Related Compounds
J. Szmuszkovicz, E. M. Glenn, R. V. Heinzelman, J. B. Hester, and G. A. Youngdale
pp 527 - 536; DOI:
10.1021/jm00322a020
PDF
Structure-Activity Studies with the Selective Rat Toxicant Norbormide
G. I. Poos, R. J. Mohrbacher, E. L. Carson, V. Paragamian, B. M. Puma, C. R. Rasmussen, and A. P. Roszkowski
pp 537 - 540; DOI:
10.1021/jm00322a021
PDF
2-Sulfanilamido-5-methoxy-1,3,4-thiadiazole and Related Compounds
M. L. Sassiver and R. G. Shepherd
pp 541 - 545; DOI:
10.1021/jm00322a022
PDF
Novel Broad-Spectrum Anthelmintics. Tetramisole1 and Related Derivatives of 6-Arylimidazo[2,1-b]thiazole
Alfons H. M. Raeymaekers, Fernand T. N. Allewijn, Jan Vandenberk, Paul J. A. Demoen, Theo T. T. Van Offenwert, and Paul A. J. Janssen
pp 545 - 551; DOI:
10.1021/jm00322a023
PDF
Semisynthetic Penicillins. III. Heterocyclic Penicillins
A. W. Chow, N. M. Hall, J. R. E. Hoover, M. M. Dolan, and R. J. Ferlauto
pp 551 - 555; DOI:
10.1021/jm00322a024
PDF
Activity of a Series of Piperdines against Haemonchus contortus Larvae
J. H. Arundel, T. C. Somers, and G. J. Handley
pp 555 - 558; DOI:
10.1021/jm00322a025
PDF
Potential Antiradiation Drugs. III.1 2-Amino-2-alkyl-1,3-propanedithiols and 3-Amino-4-mercapto-1-butanol2
G. Richard Handrick and Edward R. Atkinson
pp 558 - 562; DOI:
10.1021/jm00322a026
PDF
Modification of Radioprotective 2-Aminoethanethiol Derivatives by N,N′-Polymethylene Bridging
James R. Piper, Carl R. Stringfellow, and Thomas P. Johnston
pp 563 - 566; DOI:
10.1021/jm00322a027
PDF
Nucleosides. XXXIII. N4-Acylated 5-Fluorocytosines and a Direct Synthesis of 5-Fluoro-2′-deoxycytidine
R. Duschinsky, T. Gabriel, M. Hoffer, J. Berger, E. Titsworth, E. Grunberg, J. H. Burchenal, and J. J. Fox
pp 566 - 572; DOI:
10.1021/jm00322a028
PDF
Pyrimidines. XVIII. 2,4-Diamino-5-nitro-6-arylaminopyrimidines. Nitration Study of 2,4-Diamino-6-chloropyrimidine and a Literature Correction
Darrell E. O'Brien, C. C. Cheng, and Wolfgang Pfleiderer
pp 573 - 575; DOI:
10.1021/jm00322a029
PDF
Enzyme Inhibitors. XIII. The Synthesis of an Active-Site-Directed Irreversible Inhibitor of Adenosine Deaminase
Howard J. Schaeffer and Eugene Odin
pp 576 - 581; DOI:
10.1021/jm00322a030
PDF
Boron Hydride Anions. I. Nitrogen Mustards
F. Haslinger, A. H. Soloway, and D. N. Butler
pp 581 - 584; DOI:
10.1021/jm00322a031
PDF
The Carcinostatic Activity of Thiosemicarbazones of Formyl Heteroaromatic Compounds.1 III. Primary Correlation
Frederic A. French and Erwin J. Blanz
pp 585 - 589; DOI:
10.1021/jm00322a032
PDF
Synthesis of a Pyrimidine Analog of Tetrahydrohomofolic Acid
George L. Tong, William W. Lee, and Leon Goodman
pp 590 - 593; DOI:
10.1021/jm00322a033
PDF
Derivatives of Fluorene. XXII.1a,b Nitrogen Mustards. II1c
T. Lloyd Fletcher, William H. Wetzel, and Moses J. Namkung
pp 593 - 598; DOI:
10.1021/jm00322a034
PDF
Synthesis of Potential Antineoplastic Agents. XIV. Some 2-Substituted 2,3-Dihydro-1H-perimidines
William Wasulko, Adria Catala Noble, and Frank D. Popp
pp 599 - 601; DOI:
10.1021/jm00322a035
PDF
The Preparation and Pharmacology of Some 1,4-Dimethylestratrienes
Leland J. Chinn
pp 602 - 603; DOI:
10.1021/jm00322a036
PDF
Synthesis and Pharmacological Evaluation of α-Substituted 1-Naphthylacetic Acids
Gianfranco Pala, Tiberio Bruzzese, Ernesta Marazzi-Uberti, and Germano Coppi
pp 603 - 605; DOI:
10.1021/jm00322a037
PDF
Effect of Organic Compounds on Reproductive Processes. II. Alkylating Agents Derived from Various α,ω-Alkylenediols
W. A. Skinner, J. Hayford, T. E. Shellenberger, and W. T. Colwell
pp 605 - 607; DOI:
10.1021/jm00322a038
PDF
Nitrogen Mustard Type Derivatives of Thiophene and Benzo[b]thiophene
David A. Shirley and George R. Bell
pp 607 - 609; DOI:
10.1021/jm00322a039
PDF
Studies on Methylglyoxal Bis(guanylhydrazone)1 Analogs. V. Methylglyoxal Guanylhydrazone Thiosemicarbazones and Related Compounds2
Eugene G. Podrebarac and C. C. Cheng
pp 609 - 610; DOI:
10.1021/jm00322a040
PDF
Some Congeners and Analogs of Dipyridamole
Daniel Kaminsky, Wilson B. Lutz, and Sam Lazarus
pp 610 - 612; DOI:
10.1021/jm00322a041
PDF
Synthesis and Pharmacological Activity of a Series of 2-Substituted Pyridazinones
Julian G. Michels, George C. Wright, and Gabriel Gever
pp 612 - 615; DOI:
10.1021/jm00322a042
PDF
3-Aminopiperidones.1a II. 2-(N,N-Diethylamino)-2-phenylglutarimide1b,c
V. L. Narayanan and C. F. Martin
pp 615 - 617; DOI:
10.1021/jm00322a043
PDF
Antiviral Compounds. XIII. Aminoacethydrazones of Aromatic α-Ketoaldehydes
E. Massarani, D. Nardi, L. Degen, and M. J. Magistretti
pp 617 - 618; DOI:
10.1021/jm00322a044
PDF
Potential Antimicrobial Agents. Bromo Compounds of Eugenol
Noël J. de Souza, A. N. Kothare, and V. V. Nadkarny
pp 618 - 620; DOI:
10.1021/jm00322a045
PDF
Arylazo Derivatives of Pyridoxine
A. R. Katritzky, H. Z. Kucharska, M. J. Tucker, and H. M. Wuest
pp 620 - 622; DOI:
10.1021/jm00322a046
PDF
Studies on Latent Derivatives of Aminoethanethiols as Potentially Selective Cytoprotectants. V. Syntheses of S-(2-Aminoethyl) Methyl Hydrogen Phosphorothioate
Kurt Pollack and Orrie M. Friedman
pp 622 - 623; DOI:
10.1021/jm00322a047
PDF
Antiacetylcholinesterase Activity of O,O-Diethyl-S-(acetylphenylurea)dithiophosphoric Acid Esters
A. K. Sen Gupta, R. C. Srivastava, and Surendra S. Parmar
pp 623 - 623; DOI:
10.1021/jm00322a048
PDF
Synthesis of Varied Heterocyclic and Substituted Aryl Alkyl Secondary Amines, Related Schiff Bases, and Amides
Gordon N. Walker and Miriam Ann Klett
pp 624 - 630; DOI:
10.1021/jm00322a049
PDF
Some 3,4,5-Trimethoxphenyl Analogs of Antihistamines
Louis T. DiFazio and Pierre F. Smith
pp 631 - 632; DOI:
10.1021/jm00322a050
PDF
O-Diethyl Phosphoryl Esters of Quaternary and Tertiary Aminophenols
Sara Ginsburg, Richard J. Kitz, and Irwin B. Wilson
pp 632 - 633; DOI:
10.1021/jm00322a051
PDF
6,12-Diphenyldibenzo[b,f][1,5]diazocines
W. Metlesics, T. Resnick, G. Silverman, R. Tavares, and L. H. Sternbach
pp 633 - 634; DOI:
10.1021/jm00322a052
PDF
The Preparation of 5-Substituted 5-(2-Naphthyl)hydantoins as Potential Anticonvulsants
Ronald D. Garrett and Henry R. Henze
pp 634 - 635; DOI:
10.1021/jm00322a053
PDF
Heterocycles. II.1 Synthesis of 3-Carbomethoxy-3-methyl-7,8-benzothiochromanone
Tosio Moriwake
pp 635 - 635; DOI:
10.1021/jm00322a054
PDF
Synthesis of Some 3-Arylacetyl- and 1,3-Di(arylacetyl)indoles
Thomas E. Young and Michael F. Mizianty
pp 635 - 637; DOI:
10.1021/jm00322a055
PDF
Derivatives of 4-Phenyl-Δβ,γ-butenoides
Price Truitt and Sharon G. Truitt
pp 637 - 638; DOI:
10.1021/jm00322a056
PDF
Synthesis of 1,1′-Trimethylene-4,4′-Substituted Pyridinium and 1,3′-Halopropyl-4-Substituted Pyridinium Compounds
Clinton N. Corder and James L. Way
pp 638 - 640; DOI:
10.1021/jm00322a057
PDF
Preparation of 4-Iodoacetamido-1-naphthol as a Histochemical Reagent for Sulfhydryl Groups
K. C. Tsou and Arnold M. Seligman
pp 640 - 641; DOI:
10.1021/jm00322a058
PDF
cis-4-Aminomethylcyclohexanecarboxylic Acid
Walter E. Meyer
pp 641 - 641; DOI:
10.1021/jm00322a059
PDF
Some Solvatochromic Chelating Agents
A. Mueller and J. P. Phillips
pp 641 - 642; DOI:
10.1021/jm00322a060
PDF
Some Hydrazones of 5-Phenyl-2,4-thiazolidinedione
Aleksey A. Sirotenko and Peter A. Ciavarri
pp 642 - 643; DOI:
10.1021/jm00322a061
PDF
The Chemistry of Samandarine Model Compounds
H. Franke and R. Partch
pp 643 - 644; DOI:
10.1021/jm00322a062
PDF
Clinical Pathology.
Alfred Burger
pp 644 - 644; DOI:
10.1021/jm00322a063
PDF
Peptides and Amino Acids.
Alfred Burger
pp 644 - 644; DOI:
10.1021/jm00322a064
PDF

Issue 5


Synthesis of 1-L-Penicillamine-oxytocin, 1-D-Penicillamine-oxytocin, and 1-Deaminopenicillamine-oxytocin, Potent Inhibitors of the Oxytocic Response of Oxytocin
Horst Schulz and Vincent Du Vigneaud
pp 647 - 650; DOI:
10.1021/jm00323a001
PDF
Relationship between Configuration and Adrenergic β-Receptor Blocking Activity of Optical Isomers of 1-(4-Nitrophenyl)-2-isopropylaminoethanol (INPEA)
Luigi Almirante and Walter Murmann
pp 650 - 653; DOI:
10.1021/jm00323a002
PDF
Spiranes. XII. Azaspiranylalkylphenothiazines
Charles H. Grogan, Rafael Kelly, and Leonard M. Rice
pp 654 - 656; DOI:
10.1021/jm00323a003
PDF
Benzocyclobutene Derivatives. Oximes with Muscle Relaxant Characteristics
Joseph A. Skorcz, John T. Suh, Claude I. Judd, Murray Finkelstein, and Alvin C. Conway
pp 656 - 659; DOI:
10.1021/jm00323a004
PDF
Imidazolecarboxhydrazides. I. Chemistry and Biological Evaluation
Jay Nematollahi, Wallace Guess, and John Autian
pp 660 - 664; DOI:
10.1021/jm00323a005
PDF
3-Phenylcinnolines. I. Some Reactions and Derivatives of 3-Phenylcinnoline-4-carboxylic Acids
Harman S. Lowrie
pp 664 - 669; DOI:
10.1021/jm00323a006
PDF
3-Phenylcinnolines. II.1 The Preparation of 4-Amino Derivatives
Harman S. Lowrie
pp 670 - 675; DOI:
10.1021/jm00323a007
PDF
N-Monoalkyl-β-alkylcinnamamides as Sedatives
E. Van Heyningen, C. N. Brown, F. José, J. K. Henderson, and P. Stark
pp 675 - 681; DOI:
10.1021/jm00323a008
PDF
Nonclassical and Other sp2-Hybridized Steroids. Methano-, Spirocyclopropyl-, and Methylenepregnane Derivatives
Manfred E. Wolff, Winston Ho, and Masao Honjoh
pp 682 - 685; DOI:
10.1021/jm00323a009
PDF
Anabolic Agents. 19-Nor- and 19-Substituted 5α-Androst-2-ene Derivatives
R. E. Counsell, G. W. Adelstein, P. D. Klimstra, and B. Smith
pp 685 - 689; DOI:
10.1021/jm00323a010
PDF
Chemical and Biological Properties of Some 17-Substituted Estradiol Derivatives
R. E. Counsell, P. D. Klimstra, R. L. Elton, and E. F. Nutting
pp 689 - 692; DOI:
10.1021/jm00323a011
PDF
Anabolic Agents. 2,3-Epithioandrostane Derivatives
P. D. Klimstra, E. F. Nutting, and R. E. Counsell
pp 693 - 697; DOI:
10.1021/jm00323a012
PDF
Pteridinecarboxamide Diuretics. I. Reaction of 4,6-Diamino-5-nitrosopyrimidines with Substituted Malonamides
T. S. Osdene, Arthur A. Santilli, Lee E. McCardle, and Marvin E. Rosenthale
pp 697 - 701; DOI:
10.1021/jm00323a013
PDF
Chemistry of Dichloromaleimides. II.1 The Synthesis and Pharmacology of 1-(2-Arylamino-3-maleimidyl)pyridinium Salts
Marvin J. Karten and Allan Schwinn
pp 702 - 703; DOI:
10.1021/jm00323a014
PDF
Synthesis of Potential Antineoplastic Agents. XV. Some 1,4-Bisamides of 1,2,3,4-Tetrahydroquinoxaline
Peter Schuyler, Frank D. Popp, Adria Catala Noble, Dru W. Alwani, and Barry R. Masters
pp 704 - 707; DOI:
10.1021/jm00323a015
PDF
Hypoglycemic Activity and Pharmacological Picture of 4-(1-Naphthyl)butylamine Derivatives
Silvano Casadio, Tiberio Bruzzese, Gianfranco Pala, Germano Coppi, and Carla Turba
pp 707 - 714; DOI:
10.1021/jm00323a016
PDF
Fluorinated Pyrimidines. XXVIII. The Synthesis of 5-Trifluoromethyl-6-azauracil and 5-Trifluoromethyl-6-aza-2′-deoxyuridine
Anthony Dipple and Charles Heidelberger
pp 715 - 718; DOI:
10.1021/jm00323a017
PDF
o-Methoxy Derivatives of the Carcinogen, N-2-Fluorenylacetamide. Potential Latent Biological Arylating Agents
H. T. Nagasawa and H. R. Gutmann
pp 719 - 725; DOI:
10.1021/jm00323a018
PDF
Potential Carcinolytic Agents.1 IV. Diazoamino Mustards
Zinon B. Papanastassiou, Robert J. Bruni, Edward White, and Philip L. Levins
pp 725 - 729; DOI:
10.1021/jm00323a019
PDF
Tumor Localizing Agents. Radioactive Iodofluorenaminesulfonic Acids
Krishna C. Agrawal and Francis E. Ray
pp 729 - 732; DOI:
10.1021/jm00323a020
PDF
Triazeno-v-triazole-4-carboxamides. Synthesis and Antitumor Evaluation
Y. Fulmer Shealy and C. Allen O'Dell
pp 733 - 737; DOI:
10.1021/jm00323a021
PDF
Some Nuclear-Substituted Derivatives of α-Methyldopa
Anilkumar Parulkar, Alfred Burger, and Dorothea Aures
pp 738 - 741; DOI:
10.1021/jm00323a022
PDF
Chemistry of Cephalosporin Antibiotics. V.1 Amides and Esters of Cephalothin2
Robert R. Chauvette and Edwin H. Flynn
pp 741 - 745; DOI:
10.1021/jm00323a023
PDF
Chemistry of Cephalosporin Antibiotics. VII. Synthesis of Cephaloglycin1 and Some Homologs
John L. Spencer, Edwin H. Flynn, Roger W. Roeske, Fai Y. Siu, and Robert R. Chauvette
pp 746 - 750; DOI:
10.1021/jm00323a024
PDF
Antiparasitic Agents. I. 2-(Nitro-heterocyclic) Benzimidazoles, Benzoxazoles, and Benzothiazoles
G. L. Dunn, P. Actor, and V. J. DiPasquo
pp 751 - 753; DOI:
10.1021/jm00323a025
PDF
5,6-Dihydro-4H-1,3,4-oxadiazines. V. Base-Catalyzed Cyclodehydrohalogenation of 2-(β-Chloroalkyl)carboxylic Acid Hydrazides
Donald L. Trepanier, Vilmars Sprancmanis, and John N. Eble
pp 753 - 758; DOI:
10.1021/jm00323a026
PDF
The Chemical, Spectral, and Biological Properties of Monomethine Cyanine Dyes Containing 1,3-Benzoxazine and Quinazoline Nuclei
Richard W. J. Carney, Janice Wojtkunski, Edward A. Konopka, and George DeStevens
pp 758 - 762; DOI:
10.1021/jm00323a027
PDF
Tremorine-Antagonistic Cyclic Ketals. The Reactions of Epoxy Ethers with Ethylene Chlorohydrin
H. L. Johnson, A. R. Patel, and J. F. Oneto
pp 762 - 765; DOI:
10.1021/jm00323a028
PDF
Spiranes. XI. Spiro Derivatives from 7-Methoxy-β-tetralone
Leonard M. Rice, Kenneth R. Scott, and Charles H. Grogan
pp 765 - 766; DOI:
10.1021/jm00323a029
PDF
1-Amino-2-(4-imidazolyl)cyclopropanecarboxylic Acid
Robert A. Pages and Alfred Burger
pp 766 - 768; DOI:
10.1021/jm00323a030
PDF
Central Nervous System Depressant Imides of Cyclobutanecarboxylic Acid
Robert T. Buckler and Charles H. Jarboe
pp 768 - 770; DOI:
10.1021/jm00323a031
PDF
Some 3-Arylaminoquinoxaline-2-carboxylic Acids
Joseph G. Lombardino
pp 770 - 771; DOI:
10.1021/jm00323a032
PDF
Total Synthesis of Unsaturated Phosphatidylserine Using the N-4-Chlorobutyroyl Protecting Group
D. L. Turner, M. J. Silver, and E. Baczynski
pp 771 - 772; DOI:
10.1021/jm00323a033
PDF
1,3,2-Diazaphosphorine 2-Oxides. III.1 Preparation and Biological Evaluation of Some 1,3-Bis(aralkyl)-2-halo-1,3,2-diazaphosphorine 2-Oxides and Related Compounds2
John H. Billman, John L. Meisenheimer, and Ralph F. May
pp 772 - 774; DOI:
10.1021/jm00323a034
PDF
Synthesis of Potential Antineoplastic Agents. XVI. Cyano Derivatives of 1,2,3,4-Tetrahydroquinoxaline and Related Compounds
Peter Schuyler, Frank D. Popp, and Adria Catala Noble
pp 774 - 776; DOI:
10.1021/jm00323a035
PDF
Carcinostatic Sulfonic Acid Esters of Butyne-and Butane-1,4-diols
Robert A. Earl and Robert E. Harmon
pp 776 - 778; DOI:
10.1021/jm00323a036
PDF
Synthesis of N-Monosubstituted 2-Mercaptoethylamines with Thioureido Substituents
O. LeRoy Salerni and Robert N. Clark
pp 778 - 779; DOI:
10.1021/jm00323a037
PDF
Some Bridgehead-Substituted Tetrahydroacenaphthenones
E. Campaigne, Wendell L. Roelofs, and Richard F. Weddleton
pp 779 - 781; DOI:
10.1021/jm00323a038
PDF
The Synthesis of Some 2,3-Epithio-5α-pregnanes
P. D. Klimstra
pp 781 - 782; DOI:
10.1021/jm00323a039
PDF
Totally Synthetic Steroid Hormones. X.1 Some (±)-13β-Ethyl-7α-methylgonane Derivatives
G. C. Buzby, C. R. Walk, and Herchel Smith
pp 782 - 784; DOI:
10.1021/jm00323a040
PDF
3-Phenylcinnolines. III.1 Derivatives of Hydroxy-3-phenylcinnolines
Harman S. Lowrie
pp 784 - 786; DOI:
10.1021/jm00323a041
PDF
Structure-Hypoglycemic Activity Relationships in 1-Naphthylalkylamines
Gianfranco Pala, Silvano Casadio, Tiberio Bruzzese, and Germano Coppi
pp 786 - 788; DOI:
10.1021/jm00323a042
PDF
Substituted 2-(5-Nitro-2-furyl)benzimidazoles
P. M. G. Bavin
pp 788 - 790; DOI:
10.1021/jm00323a043
PDF
The Synthesis of Tertiary Arylalkylamines from Aryl Grignard Reagents
P. M. G. Bavin, C. R. Ganellin, J. M. Loynes, P. D. Miles, and H. F. Ridley
pp 790 - 791; DOI:
10.1021/jm00323a044
PDF
D-Arabinose and 2-Deoxy-D-ribose Derivatives
Paul F. Wiley and E. Louis Caron
pp 791 - 792; DOI:
10.1021/jm00323a045
PDF
Carboranes. II. An Analog of 1,4-(Dimethanesulfonoxy)butane
F. Haslinger and A. H. Soloway
pp 792 - 792; DOI:
10.1021/jm00323a046
PDF
Some Hydrazine Derivatives of (4-Biphenylyl)glyoxal
G. J. Durant, H. F. Ridley, and R. G. W. Spickett
pp 792 - 793; DOI:
10.1021/jm00323a047
PDF
Synthesis of 1-Benzyltryptamine
Asher Kalir and Stephen Szara
pp 793 - 794; DOI:
10.1021/jm00323a048
PDF
Survey of European Nonconventional Chemical Notation Systems.
Paul N. Craig
pp 794 - 794; DOI:
10.1021/jm00323a049
PDF
Clinical Pharmacology (Dilling).
Alfred Burger
pp 794 - 794; DOI:
10.1021/jm00323a050
PDF

Issue 6


The Analysis of Physiological Activity of Substituted Phenols with Substituent Constants
Toshio Fujita
pp 797 - 803; DOI:
10.1021/jm00324a001
PDF
Antispasmodic ortho-Substituted Phenoxyalkylamines
K. Rubinstein, N. Elming, J. Fakstorp, K. Hermansen, J. G. A. Pedersen, and T. Natvig Jacobsen
pp 804 - 809; DOI:
10.1021/jm00324a002
PDF
Serotonin Inhibitors. III.1 Compounds Related to 2′-(3-Dimethylaminopropylthio)cinnamanilide2,3
John Krapcho and Chester F. Turk
pp 809 - 812; DOI:
10.1021/jm00324a003
PDF
Some Cardiovascular Effects of a Series of Aryloxyalkylamines. II
J. Augstein, W. C. Austin, C. A. Bartram, and R. J. Boscott
pp 812 - 818; DOI:
10.1021/jm00324a004
PDF
Some Indole and Benzo[b]thiophene Derivates. Synthesis and Pharmacology
N. B. Chapman, K. Clarke, and B. Iddon
pp 819 - 823; DOI:
10.1021/jm00324a005
PDF
Structure-Activity Relationship in a Series of Adrenergic β-Blocking Agents Related to 1-(4-Nitrophenyl)-1-hydroxy-2-isopropylaminoethane (INPEA)
P. Somani, Romeo T. Bachand, W. Murmann, and L. Almirante
pp 823 - 825; DOI:
10.1021/jm00324a006
PDF
The Interaction of Pyridoxal Phosphate with Tyrosine Analogs
Nicolas Zenker
pp 826 - 828; DOI:
10.1021/jm00324a007
PDF
2-Aminotyrosine, an Analog of Tyrosine
Alvie L. Davis, John W. Zaun, Perry C. Reeves, Robert L. Hance, and Tommy J. McCord
pp 828 - 830; DOI:
10.1021/jm00324a008
PDF
N-Methyl-N-2-propynyl-1-indanamine. A Potent Monoamine Oxidase Inhibitor
C. F. Huebner, Ellen M. Donoghue, A. J. Plummer, and P. A. Furness
pp 830 - 832; DOI:
10.1021/jm00324a009
PDF
Thyromimetics. VI. The Synthesis and Biological Screening of 3,5-Diiodothyroacetic and -propionic Acid Analogs
Benjamin Blank, Francis R. Pfeiffer, and Cyrus M. Greenberg
pp 832 - 834; DOI:
10.1021/jm00324a010
PDF
Phenothiazine-1-carboxylic Acids
Blaine M. Sutton and James H. Birnie
pp 835 - 837; DOI:
10.1021/jm00324a011
PDF
Histamine Releasers. II. Synthesis of a Trimer in the Formaldehyde-p-Methoxyphenethylamine Series of Histamine Releasers
Joseph I. DeGraw, Vernon H. Brown, Samuel A. Ferguson, and W. A. Skinner
pp 838 - 840; DOI:
10.1021/jm00324a012
PDF
Antiinflammatory Compounds Exhibiting Fibrinolytic Activity
Zdenek Roubal and Oldrich Nemecek
pp 840 - 842; DOI:
10.1021/jm00324a013
PDF
Acetylene Compounds of Potential Pharmacological Value. VIII. N-(4-Dialkylamino-2-butynyl)-Substituted Cyclic Imides
Richard Dahlbom, Bo Karlén, Robert George, and Donald J. Jenden
pp 843 - 846; DOI:
10.1021/jm00324a014
PDF
Studies on Morphine-like Compounds. V.1 Absolute Configuration and Conformations of Optically Active 1,2-Diphenylethylamine Derivatives
Tadashi Sasaki, Ken Kanematsu, Yojiro Tsuzuki, and Katsumi Tanaka
pp 847 - 850; DOI:
10.1021/jm00324a015
PDF
Interesting Pharmacological Properties of the Optical Isomers of α-5,9-Diethyl-2′-hydroxy-2-methyl-6,7-benzomorphan
Everette L. May and Nathan B. Eddy
pp 851 - 852; DOI:
10.1021/jm00324a016
PDF
Central Nervous System Depressants. I. 1-Aminoalkyl-3-aryl Derivatives of 2-Imidazolidinone,1a-c 2-Imidazolidinethione, and Tetrahydro-2(1H)-pyrimidinone1d
William B. Wright, Herbert J. Brabander, Robert A. Hardy, and Arnold C. Osterberg
pp 852 - 857; DOI:
10.1021/jm00324a017
PDF
Central Nervous System Depressants. II.1a 1-Aryl-3-(2-dimethylaminoethyl)-4-imidazolin-2-ones1b
William B. Wright, Herbert J. Brabander, and Robert A. Hardy
pp 858 - 860; DOI:
10.1021/jm00324a018
PDF
New Psychotropic Agents. VII.1 5H-Dibenzo[a,d]cycloheptenyl Sulfones
M. A. Davis, G. Beaulieu, J. R. Watson, and Marie-Paule Charest
pp 860 - 864; DOI:
10.1021/jm00324a019
PDF
The Preparation and Biological Activities of Some Azonino- and Azecinoindoles and Benzazecines
D. Herbst, R. Rees, G. A. Hughes, and Herchel Smith
pp 864 - 868; DOI:
10.1021/jm00324a020
PDF
Synthesis of Methylenetetrahydrofolic Acid Analogs
Mathias P. Mertes and Natubhai R. Patel
pp 868 - 873; DOI:
10.1021/jm00324a021
PDF
6-Substituted 2,4-Diamino-5-(4-carbethoxyphenylazo)pyrimidines as Potential Precursors of Tetrahydropteridine Antimetabolites
M. Chadwick, J. Hampshire, P. Hebborn, A. M. Triggle, and D. J. Triggle
pp 874 - 876; DOI:
10.1021/jm00324a022
PDF
Synthesis of Fluorinated Pyrimidines and Triazines
Mathias P. Mertes, Souheil E. Saheb, and Duane Miller
pp 876 - 881; DOI:
10.1021/jm00324a023
PDF
1,4,5,6-Tetrahydro-as-triazines. I. Sulfuric Acid Catalyzed Condensation of Nitriles and Hydrazino Alcohols
Donald L. Trepanier, Eugene R. Wagner, Guy Harris, and Allan D. Rudzik
pp 881 - 885; DOI:
10.1021/jm00324a024
PDF
Synthesis and Biological Activity of Dinucleoside Phosphates Containing 5-Fluorouracil Residues
A. Bloch, M. H. Fleysher, R. Thedford, R. J. Maue, and R. H. Hall
pp 886 - 891; DOI:
10.1021/jm00324a025
PDF
The Synthesis of Potential Anticancer Agents. XXXVI. N-Nitrosoureas.1 II. Haloalkyl Derivatives
Thomas P. Johnston, George S. McCaleb, Pamela S. Opliger, and John A. Montgomery
pp 892 - 911; DOI:
10.1021/jm00324a026
PDF
The Use of α-Amino Acids in the Synthesis of Derivatives of 2-Aminoethanethiol as Potential Antiradiation Agents
James R. Piper, Carl R. Stringfellow, and Thomas P. Johnston
pp 911 - 920; DOI:
10.1021/jm00324a027
PDF
ω-(2-Mercaptoethylamino)-1-alkanesulfonic Acid Inner Salts and Related Compounds as Potential Antiradiation Agents
Thomas P. Johnston and Carl R. Stringfellow
pp 921 - 924; DOI:
10.1021/jm00324a028
PDF
Anabolic Agents. A-Ring Oxygenated Androstane Derivatives
P. D. Klimstra, R. Zigman, and R. E. Counsell
pp 924 - 929; DOI:
10.1021/jm00324a029
PDF
Androgenic Activity of Highly Purified 5α-Androstane and 5α-Androstan-17β-ol
Ralph I. Dorfman, Wendell H. Rooks, J. Bryan Jones, and Jeffrey D. Leman
pp 930 - 931; DOI:
10.1021/jm00324a030
PDF
Preparation and Antibacterial Activity of Some Spiramycin Derivatives
R. J. Adamski, H. Heymann, S. G. Geftic, and S. S. Barkulis
pp 932 - 934; DOI:
10.1021/jm00324a031
PDF
Anticoccidial Activity in a Series of Alkyl 6,7-Dialkoxy-4-hydroxy-3-quinolinecarboxylates
Claude F. Spencer, Alan Engle, Chia-Nien Yu, Raymond C. Finch, Edward J. Watson, Frank F. Ebetino, and Cornell A. Johnson
pp 934 - 936; DOI:
10.1021/jm00324a032
PDF
Preparation of Substituted Phenethyl Alcohols and a Study of Their Bacteriostatic Action in Escherichia coli B
Ekram Z. Khafagy and J. P. Lambooy
pp 936 - 940; DOI:
10.1021/jm00324a033
PDF
The Effect of Probenecid, Phenylbutazone, and Their Analogs on the Excretion of L-Ascorbic Acid in Rats
Peter G. Dayton, Martin M. Weiss, and James M. Perel
pp 941 - 944; DOI:
10.1021/jm00324a034
PDF
Synthesis and Cytotoxicity of 4-Aminobutyrophenone Hydrochlorides and Their Substituted Pyrimidinylhydrazones
Shu-Sing Cheng, Claude Piantadosi, and J. Logan Irvin
pp 945 - 949; DOI:
10.1021/jm00324a035
PDF
Some Herbicidal Silicon Compounds
J. K. Leasure and J. L. Speier
pp 949 - 952; DOI:
10.1021/jm00324a036
PDF
1-Fluoro Steroids. II.1a 1ξ-Fluoro-5α-androst-2-en-17β-ol Acetate
Theodore J. Foell and Leland L. Smith
pp 953 - 954; DOI:
10.1021/jm00324a037
PDF
Derivatives of 1- and 2-Tetralones
George deStevens and Barbara Smolinsky
pp 954 - 957; DOI:
10.1021/jm00324a038
PDF
Ring-D-Bridge Steroid Analogs. IV.1 14α,17α-Ethenopregn-4-ene-3,20-dione2
A. J. Solo and Baldev Singh
pp 957 - 958; DOI:
10.1021/jm00324a039
PDF
Synthetic Bradykinin Analogs
Ernest Nicolaides and Marilyn Lipnik
pp 958 - 960; DOI:
10.1021/jm00324a040
PDF
2,8-Bis(substituted amino)phenothiazine 5,5-Dioxides
Ping-Lu Chien and C. C. Cheng
pp 960 - 962; DOI:
10.1021/jm00324a041
PDF
1,3-Diethyleneguanidines
Gerhard Ottmann and Haywood Hooks
pp 962 - 964; DOI:
10.1021/jm00324a042
PDF
X-Ray Media. II. Synthesis of Alkanoylbis(isophthalamic Acids) as X-Ray Contrast Agents
G. Brooke Hoey, Robert D. Rands, Philip E. Wiegert, Douglas W. Chapman, Robert L. Zey, and George B. DeLaMater
pp 964 - 966; DOI:
10.1021/jm00324a043
PDF
L-, D-, and DL-Ephedrine Phosphates
A. Larizza, G. Brancaccio, and A. Segre
pp 966 - 967; DOI:
10.1021/jm00324a044
PDF
Piperazinesulfamylurea Hypoglycemic Agent. V.
J. M. McManus
pp 967 - 968; DOI:
10.1021/jm00324a045
PDF
Some Derivatives of Cyclododecane
Alfred Burger and Charles J. Paget
pp 968 - 970; DOI:
10.1021/jm00324a046
PDF
N-Aralkylsalicylamides
Gérard Y. Paris and Clinton H. Chambers
pp 971 - 971; DOI:
10.1021/jm00324a047
PDF
Synthesis of Analogs of Bacterial Cell Wall Glycopeptides
N. C. Chaturvedi, M. C. Khosla, and Nitya Anand
pp 971 - 973; DOI:
10.1021/jm00324a048
PDF
Myclographic Agents III. Glycol Iodobenzoates
James E. Siggins and James H. Ackerman
pp 973 - 974; DOI:
10.1021/jm00324a049
PDF
Some Quinolines Containing a Cyclic Hydroxamic Acid Group
D. Noble and D. G. Wibberley
pp 974 - 976; DOI:
10.1021/jm00324a050
PDF
Metal Complexes of 2′,3′-O-Isopropylidene-6-thioinosine
Alexander Hampton and J. C. Fratantoni
pp 976 - 976; DOI:
10.1021/jm00324a051
PDF
The Interaction of Alkyl 2-Naphthyl Ketones with Isatin
Ronald D. Garrett and Henry R. Henze
pp 976 - 977; DOI:
10.1021/jm00324a052
PDF
Synthesis of Some 2,5-Diamino-4-n-butylamino-6-substituted Pyrimidines
P. L. Warner and T. J. Bardos
pp 977 - 978; DOI:
10.1021/jm00324a053
PDF
N-(2-Chloroethyl)-DL-aspartic Acid and Some Related Amino Acids
Jaime Lores Arnaiz and Juana Falszpan
pp 978 - 979; DOI:
10.1021/jm00324a054
PDF
Some Derivatives of Natural Isoflavones
Giorgio G. Ferrari and Cesare Casagrande
pp 979 - 980; DOI:
10.1021/jm00324a055
PDF
Octamethylbiguanide Perchlorate
Victor J. Bauer and S. R. Safir
pp 980 - 981; DOI:
10.1021/jm00324a056
PDF
6-Trimethylammoniopurinide
Rainer Klemm, Helmut Schulze, Martin G. Ettlinger, and Alfred R. Bader
pp 981 - 981; DOI:
10.1021/jm00324a057
PDF
Experimental Chemotherapy. Volume IV.
Alfred Burger
pp 982 - 982; DOI:
10.1021/jm00324a058
PDF
Handbook of Experimental Pharmacology. Volume XIX. 5-Hydroxytryptamine and Related Indolealkylamines.
Alfred Burger
pp 982 - 982; DOI:
10.1021/jm00324a059
PDF
Chemical Aspects of the Autonomic Nervous System.
Alfred Burger
pp 982 - 982; DOI:
10.1021/jm00324a060
PDF
Drill's Pharmacology in Medicine.
Chalmers L. Gemmill
pp 982 - 982; DOI:
10.1021/jm00324a061
PDF
The Pharmacological Basis of Therapeutics.
Chalmers L. Gemmill
pp 982 - 982; DOI:
10.1021/jm00324a062
PDF
The Pharmacological Principles of Medical Practice.
Chalmers L. Gemmill
pp 982 - 982; DOI:
10.1021/jm00324a063
PDF
An Introduction to Pharmacology.
Chalmers L. Gemmill
pp 982 - 983; DOI:
10.1021/jm00324a064
PDF
Advances in Chromatography. Volume 1.
Thomas A. Gover
pp 983 - 983; DOI:
10.1021/jm00324a065
PDF
Second Symposium on Catecholamines.
Alfred Burger
pp 983 - 983; DOI:
10.1021/jm00324a066
PDF
Methods in Drug Evaluation.
Alfred Burger
pp 983 - 983; DOI:
10.1021/jm00324a067
PDF
Impact of Basic Sciences on Medicine.
Alfred Burger
pp 984 - 984; DOI:
10.1021/jm00324a068
PDF
Handbook of Fluorescence Spectra of Aromatic Molecules.
Leonard E. Brady
pp 984 - 984; DOI:
10.1021/jm00324a069
PDF
Synthetic Methods of Organic Chemistry. Volume 20.
Alfred Burger
pp 984 - 984; DOI:
10.1021/jm00324a070
PDF
Additions and Corrections - Derivatives of Fluorene. XXI. New Halogenofluorenes. II. Further Potential Antitumor Agents.
Hsi-Lung Pan, and T. Lloyd Fletcher
pp 986 - 986; DOI:
10.1021/jm00324a071
PDF
Additions and Corrections - exo-3-Chloro-endo-6-cyano-2-norbornanone O-(Methylcarbamoyl)oxime. A New Type of Methylcarbamate with Acaricidal Activity.
Linwood K. Payne, Jr., Harry A. Stansbury, Jr., and Mathias H. J. Welden
pp 986 - 986; DOI:
10.1021/jm00324a600
PDF
Additions and Corrections - Derivatives of Fluorene. XX. Fluorofluorenes. V. New Difluoro-2-acetamidofluorenes for the Study of Carcinogenic Mechanisms.
Moses J. Namkung, T. Lloyd Fletcher, and William H. Wetzel
pp 986 - 986; DOI:
10.1021/jm00324a601
PDF
Additions and Corrections - Nucleosides. XXIX. 1-β-D-Arabinofuranosyl-5-fluorocytosine and Related Arabino Nucleosides.
Jack J. Fox, Naishun Miller, and Iris Wempen
pp 986 - 986; DOI:
10.1021/jm00324a602
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Additions and Corrections - Derivatives of Fluorene. XXII. Nitrogen Mustards. II.
T. Lloyd Fletcher, William H. Wetzel, and Moses J. Namkung
pp 986 - 986; DOI:
10.1021/jm00324a603
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Additions and Corrections - Halonitroanilides and Their Bacteriostatic Activity.
Joseph W. Baker, Ignatius Schumacher, Gerald L. Bachman, Daniel P. Roman, and Alan L. Tharp
pp 986 - 986; DOI:
10.1021/jm00324a604
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Additions and Corrections - Organic Disulfides and Related Substances. XVII. Analogsof α(2-Aminoethylio)benzoic Acid as Antiradiation Drugs.
Lamar Field, and H. K. kim
pp 986 - 986; DOI:
10.1021/jm00324a605
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